The purpose of this study is to determine the safety and tolerability of BMS-820836 after single doses
Study Type
INTERVENTIONAL
Allocation
RANDOMIZED
Purpose
TREATMENT
Masking
TRIPLE
Enrollment
68
Oral Solution, Oral, 0.025 mg, single dose, one dose
Oral Solution, Oral, 0.1 mg, single dose, one dose
Oral Solution, Oral, 0.25 mg, single dose, one dose
Local Institution
Toronto, Ontario, Canada
To assess the safety and tolerability of BMS-820836 following single-dose administration
Time frame: Within 14 days of first dose
To assess the single-dose pharmacokinetics of BMS-820836 and its N-demethylated metabolite BMS-821007
Time frame: Within 7 days of dosing
To assess the pharmacodynamics of BMS-820836
Time frame: Within 48 hours of dosing
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Oral Solution, Oral, 0.5 mg, single dose, one dose
Oral Solution, Oral, 1 mg, single dose, one dose
Oral Solution, Oral, 2 mg, single dose, one dose
Oral Solution, Oral, 3 mg, single dose, one dose
Oral Solution, Oral, 5 mg, single dose, one dose
Oral Solution, Oral, 8 mg, single dose, one dose
Oral Solution, Oral, 0 mg, single dose, one dose
Oral Solution, Oral, 3 mg, single dose, one dose
Oral Solution, Oral, 0.5 mg, single dose, one dose