Study Design : randomized, open label, single-dose, 2-way cross-over design Phase : Phase I
Study Type
INTERVENTIONAL
Allocation
RANDOMIZED
Purpose
TREATMENT
Masking
NONE
Enrollment
51
AUClast, Cmax
Time frame: Blood gathering point : 0h, 0.5h, 1h, 1.5h, 2h, 3h, 4h, 6h, 8h, 10h, 12h, 16h, 24h, 48h, 72h, 96h, 144h, 192h
AUCinf, Tmax, t1/2, % AUCextra
AUCinf = AUClast + Clast/λz %AUCextra = \[ (AUCinf - AUClast) / AUCinf \] ×100 t1/2 = 0.693/λz
Time frame: Blood gathering point : 0h, 0.5h, 1h, 1.5h, 2h, 3h, 4h, 6h, 8h, 10h, 12h, 16h, 24h, 48h, 72h, 96h, 144h, 192h
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